List of articles in "Drug" category - Page 42

Casokefamide (INN) also known as β-casomorphin 4027 (β-CM-4027) and [D-Ala24Tyr5]-β-casomorphin-5-amide is a peripherally-specific synthetic opioid pentapeptide with the amino acid sequence Tyr-D-Ala-Phe-D-Ala-Tyr-NH2. Derived from the β-casomorphin sequence it was designed […]

Lufuradom (INN) is a drug and benzodiazepine derivative which unlike other benzodiazepines is described as an analgesic. Similarly to its analogue tifluadom lufuradom was never marketed.

Hexapradol (INN) also referable to as α-butyl-β-hydroxy-β-phenylamphetamine is a psychostimulant drug which was never marketed.

MCOPPB is a drug which acts as a potent and selective agonist for the nociceptin receptor with a pKi of 10.07 and much weaker activity at other opioid receptors. It […]

MGS-0039 is a drug that is used in neuroscientific research which acts as a potent and selective antagonist for group II of the metabotropic glutamate receptors (mGluR2/3). It produces antidepressant […]

Ocaratuzumab (AME-133v LY2469298) is a humanized monoclonal antibody designed for the treatment of cancer and autoimmune disorders.

meta-Hydroxynorephedrine or 3-hydroxynorephedrine also known as 3β-dihydroxyamphetamine is an adrenergic drug of the amphetamine class which was patented as a vasopressor and nasal decongestant but was never marketed. It is […]

S32212 is a drug which is under preclinical investigation as a potential antidepressant medicine. It behaves as a selective combined 5-HT2C receptor inverse agonist and α2-adrenergic receptor antagonist (at all […]

Imagabalin (INN USAN; PD-332334) is a drug which acts as a ligand for the α2δ subunit of the voltage-dependent calcium channel with some selectivity for the α2δ1 subunit over α2δ2. […]

NMP-7 is a drug which acts as both a non-selective agonist of the CB1 and CB2 cannabinoid receptors and also as a blocker of T-type calcium channels the target of […]