List of articles in "Drug" category - Page 192

Lorglumide (CR-1409) is a drug which inhibits gastrointestinal motility and reduces gastric secretions acting as a cholecystokinin antagonist with fairly high selectivity for the CCKA subtype.

Ibipinabant (SLV319 BMS-646256) is a drug used in scientific research which acts as a potent and highly selective CB1 antagonist. It has potent anorectic effects in animals and was researched […]

3-((2-Methyl-4-thiazolyl)ethynyl)pyridine (MTEP) is a research drug that was developed by Merck & Co. as a selective allosteric antagonist of the metabotropic glutamate receptor subtype mGluR5.

2-Methyl-6-(phenylethynyl)pyridine (MPEP) is a research drug which was one of the first compounds found to act as a selective antagonist for the metabotropic glutamate receptor subtype mGluR5. After being originally […]

L-733060 is a drug developed by Merck Sharpe & Dohme which acts as an orally active non-peptide selective antagonist for the NK1 receptor binding with a Ki of 0.08nM. Only […]

Alfadolone (INN) or alphadolone is a neuroactive steroid with hypnotic effects. It is one of the components of althesin.

Tetrahydrodeoxycorticosterone (3α21-dihydroxy-5α-pregnan-20-one; THDOC) or more preferred allotetrahydroxycorticosterone is an endogenous neurosteroid. It is synthesized from the adrenal hormone deoxycorticosterone by the action of two enzymes 5α-reductase type I and 3α-hydroxysteroid […]

The drug combination clindamycin/tretinoin (trade name Ziana and Veltin) is a topical acne treatment. It combines clindamycin phosphate (1.2%) an antibiotic and tretinoin (0.025%) a retinoid. There is a generic […]

Nipecotic acid is a GABA reuptake inhibitor used in scientific research.

O-2172 is a drug developed by Organix Inc which acts as a stimulant and potent dopamine reuptake inhibitor. It is an analogue of methylphenidate where the phenyl ring has had […]