List of articles in "Drug" category - Page 112

Delmadinone (INN) is a steroidal progestin which was never marketed. An acylated derivative delmadinone acetate is used in veterinary medicine.While delmadinone is sometimes used as a synonym for delmadinone acetate […]

Quingestanol (INN BAN) is a steroidal progestin which was never marketed. An acylated derivative quingestanol acetate is used as a pharmaceutical drug.While quingestanol is sometimes used as a synonym for […]

Nomegestrol (INN) is a steroidal progestin which was never marketed. It is the parent drug of nomegestrol acetate a widely used progestogen and hormonal contraceptive.

Denaverine is an antispasmodic drug. It was developed in Germany and patented in 1974. Denaverine hydrochloride is used in veterinary medicine under the trade name Sensiblex as a muscle relaxant […]

β-Keto-Ethylbenzodioxolylbutanamine (Eutylone bk-EBDB) is a stimulant compound developed in the 1960s which has been reported as a novel designer drug.[citation needed]

WAY-208466 is a potent and highly selective full agonist of the 5-HT6 receptor. It increases GABA levels in the cerebral cortex and tolerance does not appear to occur to this […]

Elzasonan (CP-448187) is a selective 5-HT1B and 5-HT1D receptor antagonist that was under development by Pfizer for the treatment of depression but was discontinued possibly due to poor efficacy. By […]

Pruvanserin (EMD-281014 LY-2422347) is a selective 5-HT2A receptor antagonist which was under development by Eli Lilly and Company for the treatment of insomnia. It was in phase II clinical trials […]

WAY-181187 is a high affinity and selective 5-HT6 receptor full agonist. It induces robust increases in extracellular GABA levels in the frontal cortex hippocampus striatum and amygdala of rats without […]

AH-7921 is an opioid analgesic drug selective for the µ-opioid receptor having around 80% the potency of morphine when administered orally. It was discovered in the 1970s by a team […]