Fluparoxan (GR-50360) is a potent and highly selective α2-adrenergic receptor antagonist which was being investigated as an antidepressant but failed to show sufficiently significant efficacy for depression in clinical trials […]
List of articles in "Drug" category - Page 110
Ciladopa
Ciladopa (AY-27110) is a dopamine agonist with a similar chemical structure to dopamine. It was under investigation as an antiparkinsonian agent but was discontinued due to concerns of tumorogenesis in […]
Cafaminol
Cafaminol (Rhinetten Rhinoptil) is a vasoconstrictor of the xanthine class used as a nasal decongestant in Germany.
6-APDB
6-(2-Aminopropyl)-23-dihydrobenzofuran (6-APDB 4-Desoxy-MDA EMA-3) is a stimulant and entactogen drug of the phenethylamine and amphetamine classes. It is an analogue of MDA where the heterocyclic 4-position oxygen from the 34-methylenedioxy […]
Pitrazepin
Pitrazepin is a competitive GABAA and glycine receptor antagonist. It has been used to study insect and snail nervous systems in scientific research.
Norlevorphanol
Norlevorphanol is an opioid analgesic of the morphinan class. It was never marketed.
Tolgabide
Tolgabide (SL-81.0142) is a drug which was patented by Synthélabo as an anticonvulsant but was never marketed. It is an analogue of progabide and acts similarly to it as a […]
Bamaluzole
Bamaluzole is a GABA receptor agonist. It was patented as an anticonvulsant by Merck but was never marketed. There is no known scientific literature on bamaluzole and little else is […]
Guaifenesin/phenylephrine
The combination of the drugs guaifenesin and phenylephrine is a preparation against the symptoms of cold flu and allergy. Guaifenesine is an expectorant phenylephrine is a decongestant. The drug is […]
Turosteride
Turosteride (FCE-26073) is a selective inhibitor of the enzyme 5α-reductase which was under investigation by GlaxoSmithKline for the treatment of benign prostatic hyperplasia (BPH) but was never marketed. Similarly to […]