List of articles in "Drug" category - Page 82

AM-2233 is a drug that acts as a highly potent full agonist for the cannabinoid receptors with a Ki of 1.8nM at CB1 and 2.2nM at CB2 as the active […]

Org 28312 is a drug developed by Organon International which acts as a potent cannabinoid receptor full agonist at both the CB1 and CB2 receptors. It was developed with the […]

Org 28611 (SCH-900111) is a drug developed by Organon International which acts as a potent cannabinoid receptor full agonist at both the CB1 and CB2 receptors.

8-Phenyltheophylline (8-Phenyl-13-dimethylxanthine 8-PT) is a drug derived from the xanthine family which acts as a potent and selective antagonist for the adenosine receptors A1 and A2A but unlike other xanthine […]

Dapoxetine marketed as Priligy (among and other brands) is the first compound developed specially for the treatment of premature ejaculation (PE) in men 18–64 years old. Dapoxetine works by inhibiting […]

Thiopropamine is a stimulant drug which is an analogue of amphetamine where the phenyl ring has been replaced by thiophene. It has similar stimulant effects to amphetamine but with around […]

Nelotanserin (APD-125) is a drug developed by Arena Pharmaceuticals which acts as an inverse agonist on the serotonin receptor subtype 5-HT2A. It was shown to be effective and well tolerated […]

Besonprodil (CI-1041) is a drug which acts as an NMDA antagonist selective for the NR2B subunit. It is under development as a supplemental medication for Parkinson’s disease and has been […]

AM-679 is a drug that acts as a moderately potent agonist for the cannabinoid receptors with a Ki of 13.5nM at CB1 and 49.5nM at CB2.

AM-630 (6-Iodopravadoline) is a drug that acts as a potent and selective inverse agonist for the cannabinoid receptor CB2 with a Ki of 32.1nM at CB2 and 165x selectivity over […]