Tofacitinib (trade names Xeljanz and Jakvinus formerly tasocitinib CP-690550) is a drug of the janus kinase (JAK) inhibitor class discovered and developed by Pfizer. It is currently approved for the […]
List of articles in "Drug" category - Page 79
N-Desalkylflurazepam
N-Desalkylflurazepam (N-desalkyl-2-oxoquazepam) is one of the major metabolites of quazepam. It is long-acting prone to accumulation and binds unselectively to benzodiazepine receptors.
Cycrimine
Cycrimine (trade name Pagitane) is a central anticholinergic drug designed to reduce the levels of acetylcholine in the treatment of Parkinson’s disease. Its mechanism of action is to bind to […]
Perfosfamide
Perfosfamide or 4-hydroperoxycyclophosphamide (trade name Pergamid).In the live cells perfosfamide (hydroperoxycyclophosphamide) rapidly metabolizes to its redox metabolite – 4-hydroxycyclophosphamide which is also the main hepatic active metabolite of another anticancer […]
Carfenazine
Carfenazine (INN) used in the form of carphenazine maleate (USAN) is an antipsychotic agent mainly used for the treatment of chronic schizophrenia.
Benzylpenicilloyl polylysine
Benzylpenicilloyl polylysine (Pre-Pen) is used as a skin test before the administration of penicillin. It is used to detect the immunoglobulin E antibodies. The chemical structure consists of the benzylpenicilloyl […]
Benzquinamide
Benzquinamide is a discontinued antiemetic drug used in post-operative care. It was first synthesised by Pfizer in the 1960s.
Alcaftadine
Alcaftadine is used to prevent eye irritation brought on by allergic conjunctivitis. It is a H1 histamine receptor antagonist.It was approved by the U.S. Food and Drug Administration in 2010 […]
Tetrindole
Tetrindole is a tetracyclic antidepressant that functions by inhibiting monoamine oxidase A. Tetrindole has also been shown to reduce post-stressor tachycardia in rats.
Bazinaprine
Bazinaprine (SR-95191) is an experimental drug candidate. It is a monoamine oxidase inhibitor (MAOI) which is believed to be useful for the treatment of depression. The drug strongly inhibits type […]