List of articles in "Drug" category - Page 227

SB-242084 is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor. It has anxiolytic effects and enhances dopamine signalling in the limbic system […]

Lurosetron (INN) is a serotonin 5-HT3 receptor antagonist.

Eliprodil (SL-82.0715) is a drug which acts as an NMDA antagonist binding to the polyamine modulatory site. It has neuroprotective and anticonvulsant effects in animal studies but does not support […]

Lubeluzole (Prosynap) is a drug which acts as an indirect NMDA antagonist. It inhibits the release of glutamate inhibits nitric oxide synthesis and blocks calcium and sodium gated ion channels. […]

U-50488 is a drug which acts as a highly selective κ-opioid agonist but without any μ-opioid antagonist effects. It has analgesic diuretic and antitussive effects and reverses the memory impairment […]

HZ-2 is a drug which acts as a highly selective κ-opioid agonist. It is a potent analgesic with around the same potency as morphine with a long duration of action […]

Xanomeline (LY-246708; Lumeron Memcor) is a muscarinic acetylcholine receptor agonist with reasonable selectivity for the M1 and M4 subtypes though it is also known to act as a M5 receptor […]

Spiradoline (U-62066) is a drug which acts as a highly selective κ-opioid agonist. It has analgesic diuretic and antitussive effects and produces subjective effects in animals similar to those of […]

Methoxyphenamine (trade names ASMI Euspirol Orthoxine Ortodrinex Proasma) also known as 2-methoxy-N-methylamphetamine (OMMA) is a β-adrenergic receptor agonist of the amphetamine class used as a bronchodilator.

LY-404187 (or LY404187) is an ampakine (or AMPA receptor potentiator) developed by Eli Lilly and Company. It is a member of the biarylpropylsulfonamide class of ampakines.LY-404187 has been demonstrated to […]