Delucemine (NPS-1506) is a drug which acts as an NMDA antagonist and a serotonin reuptake inhibitor and has neuroprotective effects. It was originally investigated for the treatment of stroke but […]
List of articles in "Drug" category - Page 225
Nemonapride
Nemonapride (Emilace) is an atypical antipsychotic approved in Japan for the treatment of schizophrenia. It was launched by Yamanouchi in 1991. Nemonapride acts as a D2 and D3 receptor antagonist […]
Fasudil
Fasudil hydrochloride (INN) is a potent Rho-kinase inhibitor and vasodilator. Since it was discovered it has been used for the treatment of cerebral vasospasm which is often due to subarachnoid […]
Falecalcitriol
Falecalcitriol (INN) is an analog of calcitriol. It has a higher potency both in vivo and in vitro systems and longer duration of action in vivo.
Sofalcone
Sofalcone (INN) is an oral gastrointestinal medication. It is a synthetic derivative of sophoradin a chalconoid a type of natural phenol found in Sophora tonkinensis (or Sophora subprostrata) a herb […]
Tilisolol
Tilisolol (INN trade name Selecal) is a beta blocker.
Binospirone
Binospirone (MDL-73005-EF) is a drug which acts as a partial agonist at 5-HT1A somatodendritic autoreceptors but as an antagonist at postsynaptic 5-HT1A receptors. It has anxiolytic effects.
Sarpogrelate
Sarpogrelate (Anplag MCI-9042 LS-187118) is a drug which acts as an antagonist at the 5HT2A and 5-HT2B receptors. It blocks serotonin-induced platelet aggregation and has applications in the treatment of […]
Deramciclane
Deramciclane (EGIS-3886) is a drug which acts as an antagonist at the 5-HT2A receptor as an inverse agonist at the 5-HT2C receptor and as a GABA reuptake inhibitor.In 2003 Orion […]
Bemesetron
Bemesetron (MDL-72222) is a drug which acts as an antagonist at the 5HT3 receptor. It has antiemetic effects comparable to metoclopramide however it is not used clinically instead its main […]