Tags: Drug.

Picenadol (LY-97435) is a 4-phenylpiperidine derivative that is an opioid analgesic drug developed by Eli Lilly in the 1970s.Picenadol is an effective analgesic with similar efficacy to pethidine (meperidine). It has been investigated for some applications such as obstetrics and dentistry but never commercialised.It is unusual in that one enantiomer is a pure μ-opioid agonist while the other is an antagonist. The (3R4R) isomer is the agonist while (3S4S) is antagonist.

Picenadol.svg
ATC prefix
none
CAS number
79201-85-7
FDA UNII code
TV3535QWTJ
IUPAC name
3-(13-dimethyl-4-propylpiperidin-4-yl)phenol
PubChem
53077

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