Tags: Drug.

Moxazocine (BL-4566) is an opioid analgesic of the benzomorphan family which was never marketed. It acts as a partial agonist or mixed agonist/antagonist of the opioid receptors and binds preferentially to the κ-opioid receptor. Despite its failure to reach the market clinical studies demonstrated moxazocine to be approximately 10x as potent by weight as morphine as an analgesic.

Moxazocine_structure.svg
CAS number
58239-89-7
IUPAC name
(1S9R13S)-10-(cyclopropylmethyl)-13-methoxy-1-methyl-10-azatricyclo[7.3.1.027]trideca-246-trien-4-ol

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