Isamoltane (CGP-361A) is a drug used in scientific research. It acts as an antagonist at the β-adrenergic 5-HT1A and 5-HT1B receptors. It has about five times the potency for the 5-HT1B receptor (21 nmol/l) over the 5-HT1A receptor (112 nmol/l). It has anxiolytic effects in rodents.
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