3β-(p-Fluorobenzoyloxy)tropane (8-Methyl-8-azabicyclo[3.2.1]oct-3-yl 4-fluorobenzoic acid ester 4-fluorotropacocaine 3-Pseudotropyl-4-fluorobenzoate 3-pseudotropyl-4-fluorobenzoate pFBT) is a tropane derivative drug which acts as a local anaesthetic having around 30% the stimulant potency of cocaine but around […]
List of articles in "Drug" category - Page 220
Bopindolol
Bopindolol (INN) is a beta blocker. It is an ester which acts as a prodrug for pindolol.
Fadrozole
Fadrozole (INN marketed as Afema by Novartis) is an aromatase inhibitor that has been introduced in Japan for the treatment of breast cancer.It is selective.
Iodocyanopindolol
Iodocyanopindolol (INN) is a drug related to pindolol which acts as both a β1 adrenoreceptor antagonist and a 5-HT1A receptor antagonist. Its 125I radiolabelled derivative has been widely used in […]
Cyanopindolol
Cyanopindolol (INN) is a drug related to pindolol which acts as both a β1 adrenoreceptor antagonist and a 5-HT1A receptor antagonist. Its radiolabelled derivative iodocyanopindolol has been widely used in […]
Cianopramine
Cianopramine (Ro 11-2465) also known as 3-cyanoimipramine is a tricyclic antidepressant which is related to imipramine and acts as a serotonin reuptake inhibitor and weak serotonin receptor antagonist.
Cinanserin
Cinanserin (INN) is a 5-HT2A and 5-HT2C receptor antagonist which was discovered in the 1960s.The preparation is effective against an atypical pneumonia (SARS).
Mosapramine
Mosapramine (Cremin) is an atypical antipsychotic used in Japan. It is a potent dopamine antagonist with high affinity to the D2 D3 and D4 receptors and with moderate affinity for […]
Homochlorcyclizine
Homochlorcyclizine (INN) is an antihistamine which has been marketed in Japan since 1965. It is used in the treatment of allergies and other conditions. It also has some anticholinergic antidopaminergic […]
Mizoribine
Mizoribine (INN trade name Bredinin) is an immunosuppressive drug. The compound was first observed in Tokyo Japan in 1971. It is a natural product first isolated from the mould Eupenicillium […]