List of articles in "Drug" category - Page 183

BRL-15572 is a drug which acts as a selective antagonist for the serotonin receptor subtype 5-HT1D with around 60x selectivity over other related receptors.

CP-94253 is a drug which acts as a potent and selective serotonin 5-HT1B receptor agonist with approximately 25x and 40x selectivity over the closely related 5-HT1D and 5-HT1A receptors. It […]

Albiglutide is a glucagon-like peptide-1 agonist (GLP-1 agonist) drug under investigation by GlaxoSmithKline for treatment of type 2 diabetes.It is a dipeptidyl peptidase-4-resistant glucagon-like peptide-1 dimer fused to human albumin. […]

Pancratistatin (PST) is a natural compound initially extracted from Spider Lily a Hawaiian native plant belonging to the family Amaryllidaceae (AMD). PST has shown some strong anti cancer activities by […]

Lixivaptan (VPA-985) is a phase III pharmaceutical being developed by Cardiokine Inc. a specialty pharmaceutical company based in Philadelphia PA focused on the development of pharmaceuticals for the treatment and […]

Relcovaptan (SR-49059) is a non-peptide vasopressin receptor antagonist selective for the V1a subtype. It has shown positive initial results in tests against Raynaud’s disease dysmenorrhoea and tocolysis although it is […]

Fendiline is a calcium channel blocker.It is nonselective.

ZD6126 is a vascular-targeting agent and a prodrug of N-acetylcolchinol related to colchicine. It has shown promising results on tumors in mice.A phase I clinical trial identified gastrointestinal and cardiac […]