Cyclorphan is a hallucinogenic opioid mixed agonist–antagonist related to levorphanol discovered in the late 1960s. It is not marketed as an analgesic because of side effects related to its impact […]
List of articles in "Drug" category - Page 133
Umirolimus
Umirolimus (INN/USAN) is a macrocyclic lactone a highly lipophilic derivative of sirolimus an immunosuppressant. This drug is proprietary to Biosensors International which uses it in its own drug-eluting stents and […]
Ceftaroline fosamil
Ceftaroline fosamil (INN) /sɛfˈtærɵliːn/ brand name Teflaro in the US and Zinforo in Europe is an advanced-generation cephalosporin antibiotic. It is active against methicillin-resistant Staphylococcus aureus (MRSA) and Gram-positive bacteria. […]
Fresolimumab
Fresolimumab (GC1008) is a human monoclonal antibody and an immunomodulator. It is intended for the treatment of idiopathic pulmonary fibrosis (IPF) focal segmental glomerulosclerosis and cancer (kidney cancer and melanoma).It […]
Indium (111In) biciromab
Indium (111In) biciromab (INN trade name FibriScint developed by Centocor) was a drug targeting fibrin a protein involved in the clotting of blood. It was the Fab’ fragment of a […]
Apatinib
Apatinib also known as YN968D1 is a tyrosine kinase inhibitor that selectively inhibits the vascular endothelial growth factor receptor-2 (VEGFR2 also known as KDR). It is an orally bioavailable small […]
Binedaline
Binedaline (Ixprim) also called binodaline is a drug that was being investigated as an antidepressant in the 1980s but never marketed. It acts as a selective norepinephrine reuptake inhibitor (Ki […]
E-4031
E-4031 is an experimental class III antiarrhythmic drug that blocks potassium channels of the hERG-type.
Testosterone undecanoate
Testosterone undecanoate or testosterone undecylate is an ester of testosterone. This hormone is used in androgen replacement therapy primarily for the treatment of male hypogonadism and is currently under research […]
Tiotropium bromide
Tiotropium bromide (INN) is a long-acting 24 hour anticholinergic bronchodilator used in the management of chronic obstructive pulmonary disease (COPD). Tiotropium bromide capsules for inhalation are co-promoted by Boehringer-Ingelheim and […]