Aptazapine (CGS-7525A) is a tetracyclic antidepressant (TeCA) which was assayed in clinical trials for the treatment of depression in the 1980s but was never marketed. It is a potent α2-adrenergic […]
List of articles in "Drug" category - Page 99
Aluminium acetotartrate
Aluminium acetotartrate (or ALSOL) is an organic acid astringent and disinfectant. It is the aluminium salt of acetic acid and tartaric acid.
Anitrazafen
Anitrazifen is a drug displaying COX-2 inhibitor activity.
Tazomeline
Tazomeline (LY-287041) is a drug which acts as a non-selective muscarinic acetylcholine receptor agonist. It was in clinical trials for the treatment of cognitive dysfunction such as that seen in […]
Rogletimide
Rogletimide is a drug related in chemical structure to the sedative glutethimide but instead having pharmacological activity as a selective aromatase inhibitor similar to the related drug aminoglutethimide but with […]
Hydracarbazine
Hydracarbazine is an antihypertensive agent.
Alovudine
Alovudine is an antiviral agent.
Flucindole
Flucindole is an antipsychotic with a tricyclic structure that was never marketed. It is the 68-difluoro derivative of cyclindole.
Ciclindole
Ciclindole (INN; WIN-27147-2) also known as cyclindole (USAN) is an antipsychotic with a tricyclic structure that was never marketed. It displaces spiperone binding in vitro and elevates dopamine levels in […]
Tienopramine
Tienopramine is a tricyclic antidepressant (TCA) which was never marketed. It is an analogue of imipramine where one of the benzene rings has been replaced with a thiophene ring.