Dextrothyroxine (trade name Choloxin) saw research as an cholesterol-lowering drug but was pulled due to cardiac side-effects. It also increases hepatic lipase which in turn improves utilization of triglycerides improving […]
List of articles in "Drug" category - Page 356
U0126
U0126 is a highly selective inhibitor of both MEK1 and MEK2 a type of MAPK/ERK kinase. U0126 was found to functionally antagonize AP-1 transcriptional activity via noncompetitive inhibition of the […]
Ketazocine
Ketazocine (INN) also known as ketocyclazocine is a benzomorphan derivative used in opioid receptor research. Ketocyclazocine is an exogenous opioid that binds to the kappa opioid receptor.Activation of this receptor […]
Strontium ranelate
Strontium ranelate a strontium(II) salt of ranelic acid is a medication for osteoporosis marketed as Protelos or Protos by Servier. On 13 May 2013 Servier released a Direct Healthcare Professional […]
Diproqualone
Diproqualone is an analogue of methaqualone developed in the 1980s and marketed mainly in France and some other European countries.
Cloroqualone
Cloroqualone is an analogue of methaqualone developed in the 1980s and marketed mainly in France and some other European countries. It has sedative and antitussive properties and was sold either […]
Mecloqualone
Mecloqualone (Nubarene Casfen) is an analogue of methaqualone that was first made in 1960 and marketed mainly in France and some other European countries. It has sedative hypnotic and anxiolytic […]
Staurosporine
Staurosporine (antibiotic AM-2282 or STS) is a natural product originally isolated in 1977 from the bacterium Streptomyces staurosporeus.It was the first of over 50 alkaloids to be isolated with this […]
Rebeccamycin
Rebeccamycin is a weak topoisomerase I inhibitor isolated from Streptomyces sp. It is structurally similar to staurosporine but does not show any inhibitory activity against protein kinases. It shows significant […]
Carbetocin
Carbetocin (trade names Duratocin Pabal Lonactene) is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth particularly following Cesarean section. It is an eight amino acid […]