Ro15-4513 is a weak partial inverse agonist of the benzodiazepine class of drugs developed by Hoffmann–La Roche in the 1980s. It acts as a competitive antagonist and can therefore be […]
List of articles in "Drug" category - Page 347
Azaperone
Azaperone (Stresnil Fluoperidol) is a pyridinylpiperazine and butyrophenone neuroleptic drug with sedative and antiemetic effects which is used mainly as a tranquilizer in veterinary medicine. It is used mainly in […]
O-Desmethyltramadol
O-Desmethyltramadol (O-DT) is an opioid analgesic and the main active metabolite of tramadol.(+)-O-Desmethyltramadol is the most important metabolite of tramadol produced in the liver after tramadol is consumed.
Diprenorphine
Diprenorphine (diprenorfin Revivon M5050) is an opioid antagonist used to reverse the effects of the super-potent opioid analgesics such as etorphine and carfentanil that are used for tranquilizing large animals […]
Cobamamide
Cobamamide (AdoCbl) which is also known as adenosylcobalamin and dibencozide is along with methylcobalamin (MeCbl) one of the active forms of vitamin B12. As a nutritional supplement it is available […]
Lasofoxifene
Lasofoxifene (INN) (proposed tradename Fablyn) is a non-steroidal selective estrogen receptor modulator (SERM) which is under development by Pfizer for the prevention and treatment of osteoporosis and for the treatment […]
Motexafin gadolinium
Motexafin gadolinium (proposed tradename Xcytrin) is an inhibitor of thioredoxin reductase and ribonucleotide reductase. It has been proposed as a possible chemotherapeutic agent in the treatment of brain metastases.
Cannabigerol
Cannabigerol (CBG) is a non-psychoactive cannabinoid found in the Cannabis genus of plants. Cannabigerol is found in higher concentrations in hemp rather than in varieties of Cannabis cultivated for high […]
Ethylmethylthiambutene
Ethylmethylthiambutene (N-ethyl-N-methyl-1-methyl-33-di-2-thienylallylamine Emethibutin) is an opioid analgesic drug from the thiambutene family around 1.3x the potency of morphine. It is under international control under Schedule I of the UN Single […]
Dimethylthiambutene
Dimethylthiambutene (NN-Dimethyl-1-methyl-33-di-2-thienylallylamine Ohton Aminobutene Dimethibutin Kobaton Takaton Dimethibutin) is an opioid analgesic drug most often used in veterinary medicine in Japan and to a lesser extent in other countries in […]