Terguride (INN) is a serotonin antagonist. It is used for the treatment of hyperprolactinemia. Terguride is an oral potent antagonist of 5-HT2B and 5-HT2A (serotonin) receptors. Serotonin stimulates the proliferation […]
List of articles in "Drug" category - Page 233
Ampiroxicam
Ampiroxicam (INN) is a non-steroidal anti-inflammatory drug. It is a prodrug of piroxicam.
Lomerizine
Lomerizine (INN) is a calcium channel blocker with antimigraine properties.
Acediasulfone
Acediasulfone (INN) is an antimicrobial drug which also has antimalarial activity. It is a long-acting prodrug of dapsone which is used for treating leprosy.
Acedapsone
Acedapsone (INN) is an antimicrobial drug which also has antimalarial activity. Acedapsone or 1399 F is a diacetyl compound derived from dapsone. It was synthesized and developed in 1937 by […]
Aceburic acid
Aceburic acid (INN) is a sedative drug. It is the acetyl ester of gamma hydroxy butyrate (GHB).
U-90042
U-90042 is a sedative and hypnotic drug used in scientific research. It has similar effects to sedative-hypnotic benzodiazepine drugs but is structurally distinct and so is classed as a nonbenzodiazepine […]
Cyprodime
Cyprodime is an opioid antagonist from the morphinan family of drugs.Cyprodime is a selective opioid antagonist which blocks the μ-opioid receptor but without affecting the δ-opioid or κ-opioid receptors. This […]
Oxymorphazone
Oxymorphazone is an opioid analgesic drug related to oxymorphone. Oxymorphazone is a potent and long acting μ-opioid agonist which binds irreversibly to the receptor forming a covalent bond which prevents […]
Ditolylguanidine
Ditolylguanidine is a sigma receptor agonist. It is selective for sigma receptors but non-selective between the two sigma receptor subtypes binding to both σ1 and σ2 with equal affinity. It […]