List of articles in "Drug" category - Page 212

Octatropine methylbromide (INN) or anisotropine methylbromide (USAN) trade names Valpin Endovalpin Lytispasm and others is a muscarinic antagonist and antispasmodic. It was introduced to the U.S.

8a-Phenyldecahydroquinoline (8A-PDHQ) is a high affinity NMDA antagonist developed by a team at Parke Davis in the 1950s. It is a structural analog of Phencyclidine with slightly lower binding affinity […]

Benzthiazide (BAN/INN also known as benzothiazide; trade names Aquatag Dihydrex Diucen Edemax Exna Foven and others) is a thiazide diuretic used in the treatment of high blood pressure and edema. […]

NEFA is a moderate affinity NMDA antagonist (IC50 = 0.51 μM). It is a structural analog of phencyclidine. It was first synthesized by a team at Parke Davis in the […]

Fluvalinate (trade names include Apistan Klartan Minadox) is a synthetic pyrethroid commonly used to control varroa mites in honey bee colonies.Fluvalinate is a stable non-volatile fat-soluble compound. Fluvalinate effectiveness was […]

Ticagrelor (trade name Brilinta in the US Brilique and Possia in the EU) is a platelet aggregation inhibitor produced by AstraZeneca. The drug was approved for use in the European […]

5-I-R91150 (or R93274) is a compound that acts as a potent and selective antagonist of 5-HT2A receptors. Its main application is as its iodine-123 radiolabeled form in which it can […]

Sulfamazone (INN) is a sulfonamide antibiotic with antipyretic properties.

Iclaprim (INN) codenamed AR-100 and RO-48-2622 is a diaminopyrimidine dihydrofolate reductase (DHFR)-inhibiting extended-spectrum antibiotic active against gram positive organisms being developed for the treatment of complicated skin and soft tissue […]

Afatinib (INN; trade name Gilotrif in the US and Giotrif in Europe previously Tomtovok and Tovok) is a drug approved in much of the world (including the United States Canada […]