PipISB is a drug used in scientific research which acts as a potent and selective inverse agonist of the cannabinoid receptor CB1. It is highly selective for the CB1 receptor […]
List of articles in "Drug" category - Page 21
Butyrfentanyl
Butyr-fentanyl or butyrylfentanyl (not to be confused with 3-methylfentanyl) is a potent short-acting synthetic opioid analgesic drug. It is an analogue of fentanyl with around one quarter the potency of […]
EPI-001
EPI-001 is a BPA-derived experimental drug that is antagonistic to the intrinsically disordered amino-terminus domain of the androgen receptor. EPI-001 is being developed by the pharmaceutical company ESSA Pharma Inc […]
5-MAPB
5-MAPB (1-(benzofuran-5-yl)-N-methylpropan-2-amine) is an entactogenic drug which is structurally related to 5-APB and MDMA. It has similar effects to these drugs in humans and has been used as a recreational […]
Zicronapine
Zicronapine (zye-KRON-a-peen previously known as Lu 31-130) is an atypical antipsychotic medication currently under development by H. Lundbeck A/S. In phase II studies zicronapine did show statistical significant separation from […]
AB-PINACA
AB-PINACA is a compound that was first identified as a component of synthetic cannabis products in Japan in 2012. The pharmacological properties of this compound have not been formally studied […]
PF-03550096
PF-03550096 is a drug that acts as a potent agonist for the CB2 cannabinoid receptor with good selectivity over CB1 having Ki values of 7nM at CB2 and 1500nM at […]
AB-FUBINACA
AB-FUBINACA is a drug that acts as a potent agonist for the cannabinoid receptors with Ki values of 0.9nM at CB1 and 23.2nM at CB2. It was originally developed by […]
Zatuximab
Zatuximab (INN) is a chimeric monoclonal antibody designed for the treatment of cancer. It acts as an immunomodulator and binds to HER1.
Simtuzumab
Simtuzumab (INN; formerly GS 6624) is a humanized monoclonal antibody designed for the treatment of fibrosis. It binds to LOXL2 and acts as an immunomodulator.