List of articles in "Drug" category - Page 149

Befiradol (F-13640) is a very potent and highly selective 5-HT1A receptor full agonist. It has powerful analgesic and antiallodynic effects comparable to those of high doses of opioid painkillers but […]

Eslicarbazepine acetate (BIA 2-093) is an antiepileptic drug. It is a prodrug which is activated to eslicarbazepine (S-licarbazepine) an active metabolite of oxcarbazepine.It is being developed by Bial and will […]

CCG-4986 is a drug which is the first non-peptide compound discovered that acts as a selective inhibitor of the Regulator of G protein signalling protein subtype RGS4. Regulators of G […]

GR-127935 is a drug which acts as a selective antagonist at the serotonin receptors 5-HT1B and 5-HT1D. It has little effect when given by itself but blocks the antiaggressive effect […]

Ricasetron (BRL-46470) is a drug which acts as a selective antagonist at the serotonin 5-HT3 receptor. It has antiemetic effects as with other 5-HT3 antagonists and also has anxiolytic effects […]

SR-48692 is a drug which acts as a selective non-peptide antagonist at the neurotensin receptor NTS1 and was the first non-peptide antagonist developed for this receptor. It is used in […]

SB-215505 is a drug which acts as a potent and selective antagonist at the serotonin 5-HT2B receptor with good selectivity over the related 5-HT2A and 5-HT2C receptors. It is used […]

SHA-68 is a drug which acts as a selective non-peptide antagonist at the neuropeptide S receptor NPSR. In animal studies it has anxiogenic effects and blocks the stimulant action of […]

NGD-4715 is a drug developed by Neurogen which acts as a selective non-peptide antagonist at the melanin concentrating hormone receptor MCH1. In animal studies it has anxiolytic antidepressant and anorectic […]

SNAP-7941 is a drug used in scientific research which is a selective non-peptide antagonist at the melanin concentrating hormone receptor MCH1.