List of articles in "Drug" category - Page 142

Piperaquine is an antimalarial drug a bisquinoline first synthesised in the 1960s and used extensively in China and Indochina as prophylaxis and treatment during the next 20 years. Usage declined […]

Pyronaridine is an antimalarial drug. It was first synthesized in 1970 and has been in clinical use in China since the 1980s. It was first assayed by Adegoke and Babalola […]

L-765314 is a drug which acts as a potent and selective antagonist for the Alpha-1 adrenergic receptor subtype α1B. It has mainly been used to investigate the role of α1B […]

Sazetidine A (AMOP-H-OH) is a drug which acts as a subtype selective partial agonist at α4β2 neural nicotinic acetylcholine receptors acting as an agonist at (α4)2(β2)3 pentamers but as an […]

CP-809101 is a drug which acts as a potent and selective 5-HT2C receptor agonist. It had promising results in animal models of obesity and psychosis but associated with genotoxicity which […]

para-Chlorophenylpiperazine (pCPP) is a psychoactive drug of the phenylpiperazine class. It is relatively obscure with limited human use and produces slightly psychedelic effects.[citation needed] It has been encountered in illicit […]

JNJ-7925476 is a TRI antidepressant currently under development by Johnson & Johnson.These molecules were first prepared by Bruce E. Maryanoff et al. during the late 1970s – 1980’s. and is […]

Bardoxolone methyl (also known as “RTA 402” and “CDDO-methyl ester”) is an orally-available first-in-class synthetic triterpenoid. It is an inducer of the Nrf2 pathway which can suppress oxidative stress and […]

Olprinone (INN) is a cardiotonic agent. It has been marketed in Japan since 1996.

Metabutoxycaine marketed under the trade name Primacaine is a local anesthetic. It is used in dentistry.